TargetMol

ATX inhibitor 1

Product Code:
 
TAR-T10410
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T10410-1mg1mg£135.00
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TAR-T10410-2mg2mg£165.00
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TAR-T10410-5mg5mg£229.00
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TAR-T10410-1mL1 mL * 10 mM (in DMSO)£246.00
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TAR-T10410-10mg10mg£321.00
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TAR-T10410-25mg25mg£493.00
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TAR-T10410-50mg50mg£680.00
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TAR-T10410-100mg100mg£930.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
ATX inhibitor 1 is a potent ATX inhibitor (IC50: 1.23 nM, FS-3 and 2.18 nM, bis-pNPP).
CAS:
2225892-70-4
Formula:
C21H23Cl2N2O6P
Molecular Weight:
501.3
Pathway:
Metabolism
Purity:
0.9988
SMILES:
OP(O)(=O)Cc1ccc(NC(=O)C2CCN(CC2)C(=O)OCc2cc(Cl)cc(Cl)c2)cc1
Target:
PDE

References

1. Balupuri A, et al. Discovery and optimization of ATX inhibitors via modeling, synthesis and biological evaluation. Eur J Med Chem. 2018 Mar 25;148:397-409.