TargetMol

EBI-2511

Product Code:
 
TAR-T15194
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T15194-1mg1mg£119.00
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TAR-T15194-5mg5mg£189.00
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TAR-T15194-10mg10mg£254.00
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TAR-T15194-25mg25mg£454.00
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TAR-T15194-50mg50mg£625.00
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Quantity:
TAR-T15194-100mg100mg£867.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
EBI-2511 is a highly potent and orally active inhibitor of EZH2 (IC50: 6 nM in Pfeffiera cell lines).
CAS:
2098546-05-3
Formula:
C34H48N4O4
Molecular Weight:
576.782
Pathway:
Chromatin/Epigenetic
Purity:
0.9901
SMILES:
CCN(C1CCOCC1)c1cc2oc(cc2c(C(=O)NCc2c(C)cc(C)[nH]c2=O)c1CC)C1CCN(CC1)C(C)C
Target:
Histone Methyltransferase

References

1. Lu B, et al. Discovery of EBI-2511: A Highly Potent and Orally Active EZH2 Inhibitor for the Treatment of Non-Hodgkin's Lymphoma. ACS Med Chem Lett. 2018 Jan 29;9(2):98-102.