TargetMol

NS5806

Product Code:
 
TAR-T16348
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T16348-1mg1mg£102.00
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TAR-T16348-5mg5mg£148.00
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TAR-T16348-1mL1 mL * 10 mM (in DMSO)£169.00
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TAR-T16348-10mg10mg£195.00
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TAR-T16348-25mg25mg£281.00
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TAR-T16348-50mg50mg£383.00
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TAR-T16348-100mg100mg£531.00
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Further Information

Bioactivity:
NS5806 is an effective potassium current activator. NS5806 slows KV4.3 and KV4.2 current decay in channel complexes containing KChIP2. NS5806 enhances KV4.3/KChIP2 peak current amplitudes (EC50: 5.3 μM).
CAS:
426834-69-7
Formula:
C16H8Br2F6N6O
Molecular Weight:
574.079
Pathway:
Membrane transporter/Ion channel
Purity:
0.9963
SMILES:
FC(F)(F)c1cc(NC(=O)Nc2c(Br)cc(Br)cc2-c2nn[nH]n2)cc(c1)C(F)(F)F
Target:
Potassium Channel

References

1. Lundby A, et al. Effect of the I(to) activator NS5806 on cloned K 2. Cheng H, et al. Differential responses of rabbit ventricular and atrial transient outward current (Ito) to the Itomodulator NS5806. Physiol Rep. 2017 Mar;5(5). pii: e13172.