TargetMol

TUG-424

Product Code:
 
TAR-T17177
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T17177-1mg1mg£130.00
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TAR-T17177-1mL1 mL * 10 mM (in DMSO)£192.00
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TAR-T17177-5mg5mg£201.00
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TAR-T17177-10mg10mg£258.00
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TAR-T17177-25mg25mg£383.00
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TAR-T17177-50mg50mg£536.00
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TAR-T17177-100mg100mg£736.00
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TAR-T17177-500mg500mg£1,420.00
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Further Information

Bioactivity:
TUG-424 significantly enhances glucose-stimulated insulin secretion at 100 nM. TUG-424 is a potent and selective free fatty acid receptor 1 agonist (EC50: 32 nM).
CAS:
1082058-99-8
Formula:
C18H16O2
Molecular Weight:
264.32
Purity:
0.9977
SMILES:
O=C(O)CCC1=CC=C(C#CC=2C=CC=CC2C)C=C1

References

1. Discovery of Potent and Selective Agonists for the Free Fatty Acid Receptor 1 (FFA1/GPR40), a Potential Target for the Treatment of Type II Diabetes J. Med. Chem., 2008, 51 (22), pp 7061-7064 2. Christiansen E, et al. Discovery of potent and selective agonists for the free fatty acid receptor 1 (FFA(1)/GPR40), a potential target for the treatment of type II diabetes. J Med Chem. 2008 Nov 27;51(22):7061-4.