TargetMol

WR-99210

Product Code:
 
TAR-T17257L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
❮❯

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CodeSizePrice
TAR-T17257L-1mg1mg£184.00
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TAR-T17257L-5mg5mg£302.00
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TAR-T17257L-1mL1 mL * 10 mM (in DMSO)£330.00
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TAR-T17257L-10mg10mg£402.00
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TAR-T17257L-25mg25mg£623.00
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TAR-T17257L-50mg50mg£857.00
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Quantity:
TAR-T17257L-100mg100mg£1,131.00
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Quantity:
TAR-T17257L-500mg500mg£2,183.00
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Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
WR-99210 is a potent inhibitor of Plasmodium falciparum dihydrofolate reductase (pfDHFR), which is a major malarial drug target. It has subnanomolar potency for the wild type, double mutant and quadruple mutant dihydrofolate reductases.
CAS:
30711-93-4
Formula:
C14H19Cl4N5O2
Molecular Weight:
431.14
Purity:
0.9996
SMILES:
Cl.CC1(C)N=C(N)N=C(N)N1OCCCOc1cc(Cl)c(Cl)cc1Cl

References

1. Canfield C J , Milhous W K , Ager A L , et al. PS-15: a potent, orally active antimalarial from a new class of folic acid antagonists.[J]. American Journal of Tropical Medicine & Hygiene, 1993, 49(1):121.