TargetMol

AGI-5198

Product Code:
 
TAR-T2104
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T2104-5mg5mg£96.00
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TAR-T2104-10mg10mg£112.00
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TAR-T2104-1mL1 mL * 10 mM (in DMSO)£116.00
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TAR-T2104-50mg50mg£132.00
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TAR-T2104-100mg100mg£172.00
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This product comes from: United States.
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Further Information

Bioactivity:
AGI-5198 is a highly effective and specific inhibitor of IDH1 R132H/R132C mutants (IC50: 0.07/0.16 μM).
CAS:
1355326-35-0
Formula:
C27H31FN4O2
Molecular Weight:
462.569
Pathway:
Metabolism
Purity:
0.9923
SMILES:
Cc1nccn1CC(=O)N(C(C(=O)NC1CCCCC1)c1ccccc1C)c1cccc(F)c1
Target:
Dehydrogenase; Isocitrate Dehydrogenase (IDH)

References

1. Rohle D, et al. Science, 2013, 340(6132), 626-630.