TargetMol

Pravadoline

Product Code:
 
TAR-T21380
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T21380-1mg1mg£227.00
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TAR-T21380-5mg5mg£422.00
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TAR-T21380-10mg10mg£589.00
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TAR-T21380-25mg25mg£863.00
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TAR-T21380-50mg50mg£1,179.00
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TAR-T21380-100mg100mg£1,564.00
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Quantity:
TAR-T21380-500mg500mg£3,058.00
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Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
Pravadoline is a cannabinoid receptor agonist. Pravadoline inhibited the PGs synthesis in mouse brain and displayed antinociceptive activity in rodents subjected to a variety of thermal, chemical, and mechanical nociceptive stimuli.
CAS:
92623-83-1
Formula:
C23H26N2O3
Molecular Weight:
378.472
Pathway:
GPCR/G Protein
Purity:
0.992
SMILES:
COc1ccc(cc1)C(=O)c1c(C)n(CCN2CCOCC2)c2ccccc12
Target:
Cannabinoid Receptor

References

1. Everett RM, et al. Nephrotoxicity of pravadoline maleate (WIN 48098-6) in dogs: evidence of maleic acid-induced acute tubular necrosis. Fundam Appl Toxicol. 1993 Jul;21(1):59-65. 2. D'Ambra TE, et al. Conformationally restrained analogues of pravadoline: nanomolar potent, enantioselective, (aminoalkyl)indole agonists of the cannabinoid receptor. J Med Chem. 1992 Jan;35(1):124-35. 3. Ward SJ, et al. Pravadoline: profile in isolated tissue preparations. J Pharmacol Exp Ther. 1990 Dec;255(3):1230-9. 4. Haubrich DR, et al. Pharmacology of pravadoline: a new analgesic agent. J Pharmacol Exp Ther. 1990 Nov;255(2):511-22.