TargetMol

PIK-93

Product Code:
 
TAR-T2616
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T2616-1mg1mg£100.00
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TAR-T2616-5mg5mg£136.00
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TAR-T2616-1mL1 mL * 10 mM (in DMSO)£143.00
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TAR-T2616-10mg10mg£168.00
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TAR-T2616-25mg25mg£249.00
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TAR-T2616-50mg50mg£369.00
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Quantity:
TAR-T2616-100mg100mg£511.00
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This product comes from: United States.
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Further Information

Bioactivity:
PIK-93 is the first potent, synthetic PI4K inhibitor with IC50 of 19 nM; inhibits PI3Kα with IC50 of 39 nM.
CAS:
593960-11-3
Formula:
C14H16ClN3O4S2
Molecular Weight:
389.87
Pathway:
PI3K/Akt/mTOR signaling; DNA Damage/DNA Repair; Microbiology/Virology; Metabolism
Purity:
0.9983
SMILES:
CC(=O)Nc1nc(C)c(s1)-c1ccc(Cl)c(c1)S(=O)(=O)NCCO
Target:
ATM/ATR; DNA-PK; Virus Protease; PI3K; Carbonic Anhydrase; PI4K; mTOR; HSV

References

1. Knight ZA, Cell, 2006, 125(4), 733-747. 2. VanKeymeulen A, et al. Cell Biol. 2006, 174(3), 437-445. 3. T?th B, et al. J BiolChem, 2006, 281(47), 36369-3637 4. Monet M, et al. J BiolChem, 2012, Epub ahead of print. 5. Arita M, et al. J Virol, 2011, 85(5), 2364-2372.