TargetMol

PF-4136309

Product Code:
 
TAR-T3430
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T3430-1mg1mg£95.00
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TAR-T3430-2mg2mg£106.00
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TAR-T3430-5mg5mg£125.00
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TAR-T3430-1mL1 mL * 10 mM (in DMSO)£139.00
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TAR-T3430-10mg10mg£161.00
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Quantity:
TAR-T3430-25mg25mg£228.00
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Quantity:
TAR-T3430-50mg50mg£334.00
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Quantity:
TAR-T3430-100mg100mg£462.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
INCB8761(PF-4136309) is a specific, effective, and orally bioavailable CCR2 antagonist.
CAS:
1341224-83-6
Formula:
C29H31F3N6O3
Molecular Weight:
568.601
Pathway:
Microbiology/Virology; Immunology/Inflammation
Purity:
0.999
SMILES:
O[C@]1(CC[C@@H](CC1)N[C@H]1CCN(C1)C(=O)CNC(=O)c1cccc(c1)C(F)(F)F)c1ccc(cn1)-c1ncccn1
Target:
CCR

References

Discovery of INCB8761/PF-4136309, a Potent, Selective, and Orally Bioavailable CCR2 Antagonist By Xue, Chu-Biao; Wang, Anlai; Han, Qi; Zhang, Yingxin; Cao, Ganfeng; Feng, Hao; Huang, Taisheng; Zheng, Changsheng; Xia, Michael; Zhang, Ke; et ACS Med. Chem. Lett., 2011, 2 (12), pp 913-918