TargetMol

Sari 59-801

Product Code:
 
TAR-T34532
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T34532-1mg1mg£140.00
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TAR-T34532-5mg5mg£327.00
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TAR-T34532-1mL1 mL * 10 mM (in DMSO)£330.00
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TAR-T34532-10mg10mg£470.00
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TAR-T34532-25mg25mg£723.00
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TAR-T34532-50mg50mg£978.00
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Quantity:
TAR-T34532-100mg100mg£1,291.00
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Further Information

Bioactivity:
Sari 59-801 is a novel, orally effective hypoglycemic compound that appears to act largely by stimulation of insulin release. SARI-59-801 was more potent in producing hypoglycemia (ED25 = 47 mg/kg) than their lean littermates (ED25 = 131 mg/kg).
CAS:
80565-58-8
Formula:
C18H23N3O2
Molecular Weight:
313.401
Purity:
0.9996
SMILES:
CCc1noc(C)c1-c1[nH]c2ccccc2c1C(O)CN(C)C

References

Hanson RL, Isaacson CM. Stimulation of insulin secretion from isolated rat islets by SaRI 59-801. Relation to cAMP concentration and Ca2+ uptake. Diabetes. 1985 Jul;34(7):691-5. PubMed PMID: 2408949. Hanson RL, Isaacson CM, Boyajy LD. Stimulation of insulin secretion from isolated rat islets by SaRI 59-801. Diabetes. 1985 Jun;34(6):548-52. PubMed PMID: 3924691.