TargetMol

CFMTI

Product Code:
 
TAR-T3482
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T3482-1mg1mg£121.00
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TAR-T3482-5mg5mg£205.00
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TAR-T3482-1mL1 mL * 10 mM (in DMSO)£207.00
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TAR-T3482-10mg10mg£262.00
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TAR-T3482-25mg25mg£445.00
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TAR-T3482-50mg50mg£619.00
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Quantity:
TAR-T3482-100mg100mg£852.00
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Further Information

Bioactivity:
CFMTI is a potent and selective metabotropic glutamate receptor (mGluR) 1 allosteric antagonist (IC50: 2.6 nM). The selectivity of CFMTI to mGluR1 is higher 2000-fold than mGluR5.
CAS:
864864-17-5
Formula:
C19H16FN5O
Molecular Weight:
349.369
Pathway:
Neuroscience
Purity:
0.9861
SMILES:
Cc1c(nnn1-c1cccnc1F)-c1ccc2C(=O)N(Cc2c1)C1CC1
Target:
GluR

References

Satow A et al. Unique antipsychotic activities of the selective metabotropic glutamate receptor 1 allosteric antagonist 2-cyclopropyl-5-[1-(2-fluoro-3-pyridinyl)-5-methyl-1H-1,2,3-triazol-4-yl]-2,3-dihydro-1H-isoindol-1-one. J Pharmacol Exp Ther. 2009 Jul;330(1):179-90.