TargetMol

EST73502

Product Code:
 
TAR-T39284
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T39284-1mg1mg£195.00
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TAR-T39284-5mg5mg£325.00
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TAR-T39284-1mL1 mL * 10 mM (in DMSO)£348.00
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TAR-T39284-10mg10mg£434.00
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TAR-T39284-25mg25mg£669.00
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TAR-T39284-50mg50mg£914.00
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TAR-T39284-100mg100mg£1,187.00
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TAR-T39284-500mg500mg£2,344.00
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This product comes from: United States.
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Further Information

Bioactivity:
EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.
CAS:
2307458-82-6
Formula:
C19H27ClF2N2O2
Molecular Weight:
388.88
Pathway:
Neuroscience; GPCR/G Protein; Endocrinology/Hormones
Purity:
0.98
SMILES:
CCN1CC2(CCN(CCC3=CC(F)=CC=C3F)CC2)O[C@H](C)C1=O
Target:
Opioid Receptor

References

M?nica Garc?a, et al. Discovery of EST73502, a Dual ?-Opioid Receptor Agonist and ? 1 Receptor Antagonist Clinical Candidate for the Treatment of Pain. J Med Chem. 2020 Oct 16.