TargetMol

Asapiprant

Product Code:
 
TAR-T5386
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T5386-1mg1mg£172.00
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TAR-T5386-5mg5mg£367.00
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TAR-T5386-1mL1 mL * 10 mM (in DMSO)£431.00
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TAR-T5386-10mg10mg£497.00
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TAR-T5386-25mg25mg£760.00
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TAR-T5386-50mg50mg£1,018.00
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TAR-T5386-100mg100mg£1,340.00
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Further Information

Bioactivity:
Asapiprant (S-555739) is a potent and selective DP1 receptor antagonist (Ki: 0.44 nM). It exhibited high affinity and selectivity for the DP1 receptor.
CAS:
932372-01-5
Formula:
C24H27N3O7S
Molecular Weight:
501.55
Pathway:
GPCR/G Protein; Immunology/Inflammation
Purity:
0.9923
SMILES:
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CCN(CC1)c1ccc(-c2ncco2)c(OCC(O)=O)c1
Target:
Prostaglandin Receptor

References

Takahashi G, et al. Effect of the potent and selective DP1 receptor antagonist, asapiprant (S-555739), in animal models of allergic rhinitis and allergic asthma. Eur J Pharmacol. 2015 Oct 15;765:15-23.