TargetMol

Chaetocin

Product Code:
 
TAR-T6803
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T6803-1mL1 mL * 10 mM (in DMSO)Enquire
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TAR-T6803-2mg2mgEnquire
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TAR-T6803-1mg1mg£177.00
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TAR-T6803-5mg5mg£390.00
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TAR-T6803-10mg10mg£546.00
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This product comes from: United States.
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Further Information

Bioactivity:
Chaetocin, a natural product from Chaetomium species, is a histone methyltransferase inhibitor with IC50 of 0.8 μM, 2.5 μM and 3 μM for dSU(VAR)3-9, mouse G9a and Neurospora crassa DIM5, respectively.
CAS:
28097-03-2
Formula:
C30H28N6O6S4
Molecular Weight:
696.83
Pathway:
Microbiology/Virology; Chromatin/Epigenetic
Purity:
0.98
SMILES:
CN1C(=O)[C@@]23C[C@]4([C@H](Nc5ccccc45)N2C(=O)[C@]1(CO)SS3)[C@]12C[C@]34SS[C@](CO)(N(C)C3=O)C(=O)N4[C@H]1Nc1ccccc21
Target:
Histone Methyltransferase; Antibacterial; Antibiotic

References

Greiner D, et al. Nat Chem Biol. 2005, 1(3), 143-145. Isham CR, et al. Br J Cancer. 2012, 106(2), 314-323. Lee YM, et al. Hepatology. 2011, 53(1), 171-180.