TargetMol

Basmisanil

Product Code:
 
TAR-T7165
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T7165-2mg2mg£96.00
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Quantity:
TAR-T7165-1mL1 mL * 10 mM (in DMSO)£105.00
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TAR-T7165-5mg5mg£111.00
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TAR-T7165-10mg10mg£128.00
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Quantity:
TAR-T7165-25mg25mg£171.00
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Quantity:
TAR-T7165-50mg50mg£237.00
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Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
Basmisanil is a negative allosteric modulator/inverse agonist of GABAAα5 receptors.Formulations containing basmisanil are in clinical trials for the treatment of cognitive impairments associated with Down syndrome.
CAS:
1159600-41-5
Formula:
C21H20FN3O5S
Molecular Weight:
445.47
Pathway:
Neuroscience; Membrane transporter/Ion channel
Purity:
0.98
SMILES:
Cc1onc(c1COc1ccc(cn1)C(=O)N1CCS(=O)(=O)CC1)-c1ccc(F)cc1
Target:
GABA Receptor

References

Szepes, Anik?, Pabst-Ravot A , Storch K , et al. Stability and compatibility of Basmisanil granules co-administered with soft food[J]. International Journal of Pharmaceutics, 2018. Myers J F , Comley R A , Gunn R N . Quantification of [ 11 C]Ro15-4513 GABA A ?5 specific binding and regional selectivity in humans[J]. Journal of Cerebral Blood Flow & Metabolism, 2016, 37(6):0271678X16661339.