TargetMol

Encenicline

Product Code:
 
TAR-T7193
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T7193-1mg1mg£160.00
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TAR-T7193-2mg2mg£205.00
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TAR-T7193-5mg5mg£262.00
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TAR-T7193-1mL1 mL * 10 mM (in DMSO)£278.00
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TAR-T7193-10mg10mg£380.00
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TAR-T7193-25mg25mg£589.00
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TAR-T7193-50mg50mg£809.00
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TAR-T7193-100mg100mg£1,075.00
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This product comes from: United States.
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Further Information

Bioactivity:
Encenicline is a selective α7 nicotinic acetylcholine receptor (nAChRs) agonist in development for treating cognitive impairment in schizophrenia and Alzheimer's disease.
CAS:
550999-75-2
Formula:
C16H17ClN2OS
Molecular Weight:
320.84
Pathway:
Neuroscience
Purity:
0.98
SMILES:
Clc1cccc2cc(sc12)C(=O)N[C@H]1CN2CCC1CC2
Target:
AChR

References

Prickaerts J, van Goethem NP, Chesworth R,et al.EVP-6124, a novel and selective ?7 nicotinic acetylcholine receptor partial agonist, improves memory performance by potentiating the acetylcholine response of ?7 nicotinic acetylcholine receptors[J].Neuropharmacology. 2012 Feb;62(2):1099-110. Hayward A , Adamson L , Neill J C . Partial agonism at the ?7 nicotinic acetylcholine receptor improves attention, impulsive action and vigilance in low attentive rats[J]. European Neuropsychopharmacology, 2017, 27(4):325-335.