TargetMol

CL 218872

Product Code:
 
TAR-T8572
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T8572-1mL1 mL * 10 mM (in DMSO)£96.00
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TAR-T8572-10mg10mg£102.00
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TAR-T8572-25mg25mg£138.00
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TAR-T8572-50mg50mg£189.00
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TAR-T8572-100mg100mg£269.00
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This product comes from: United States.
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Further Information

Bioactivity:
CL 218872 is a benzodiazepine agonist displaying selectivity for α1 subunit-containing GABAA receptors (Ki values are 130, 1820, 1530, > 10000, 490 and > 10000 nM for α1, α2, α3, α4, α5 and α6-subunit containing receptors respectively). Orally active anxiolytic and anticonvulsant in vivo.
CAS:
66548-69-4
Formula:
C13H9F3N4
Molecular Weight:
278.238
Pathway:
Neuroscience; Membrane transporter/Ion channel
Purity:
0.9997
SMILES:
Cc1nnc2ccc(nn12)-c1cccc(c1)C(F)(F)F
Target:
GABA Receptor

References

Wang B , Lv K , Liu H , et al. Contribution of the ?5 GABAA receptor to the discriminative stimulus effects of propofol in rat[J]. Neuroreport, 2018:347-352.