TargetMol

MCH(human, mouse, rat)

Product Code:
 
TAR-TP1996
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-TP1996-1mg1mg£254.00
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TAR-TP1996-5mg5mg£524.00
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TAR-TP1996-10mg10mg£703.00
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TAR-TP1996-25mg25mg£1,018.00
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TAR-TP1996-50mg50mg£1,324.00
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Quantity:
TAR-TP1996-100mg100mg£1,749.00
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This product comes from: United States.
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Further Information

Bioactivity:
Potent endogenous agonist at melanin-concentration hormone (MCH) receptors (IC50 values are 0.3 and 1.5 nM and EC50 values are 3.9 and 0.1 nM at MCH1 and MCH2 receptors respectively). Increases food intake in vivo.
CAS:
128315-56-0
Formula:
C105H160N30O26S4
Molecular Weight:
2386.86
Pathway:
GPCR/G Protein; Endocrinology/Hormones
Purity:
0.9955
SMILES:
CSCC[C@H](NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@H]1CSSC[C@H](NC(=O)[C@@H]2CCCN2C(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](Cc2ccc(O)cc2)NC(=O)[C@@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCSC)NC1=O)C(C)C)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](C(C)C)C(O)=O
Target:
GPR; Melanin-concentrating Hormone Receptor (MCHR)

References

Sailer et al (2001) Identification and characterization of a second melanin-concentrating hormone receptor, MCH-2R. Proc.Natl.Acad.Sci.USA 98 7564