TargetMol

MRS-1706

Product Code:
 
TAR-T16136
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T16136-1mg1mg£95.00
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TAR-T16136-2mg2mg£106.00
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TAR-T16136-5mg5mg£128.00
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TAR-T16136-1mL1 mL * 10 mM (in DMSO)£135.00
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TAR-T16136-10mg10mg£168.00
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TAR-T16136-25mg25mg£274.00
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TAR-T16136-50mg50mg£470.00
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TAR-T16136-100mg100mg£651.00
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Further Information

Bioactivity:
MRS-1706 has Ki values of 1.39, 112, 157, and 230 nM for human A2B, A2A, A1, and A3 receptors respectively. MRS-1706 is an effective and selective adenosine A2B receptor inverse agonist.
CAS:
264622-53-9
Formula:
C27H29N5O5
Molecular Weight:
503.559
Pathway:
GPCR/G Protein; Neuroscience
Purity:
0.9795
SMILES:
CCCn1c2nc([nH]c2c(=O)n(CCC)c1=O)-c1ccc(OCC(=O)Nc2ccc(cc2)C(C)=O)cc1
Target:
Adenosine Receptor

References

1. Li Q, et al. ZM241385, DPCPX, MRS1706 are inverse agonists with different relative intrinsic efficacies on constitutively active mutants of the human adenosine A2B receptor. J Pharmacol Exp Ther. 2007 Feb;320(2):637-45. 2. Desai A, et al. Adenosine A2A receptor stimulation increases angiogenesis by down-regulating production of the antiangiogenic matrix protein thrombospondin 1. Mol Pharmacol. 2005 May;67(5):1406-13.