TargetMol

APY0201

Product Code:
 
TAR-T2061
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T2061-2mg2mg£128.00
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Quantity:
TAR-T2061-1mL1 mL * 10 mM (in DMSO)£158.00
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Quantity:
TAR-T2061-5mg5mg£158.00
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TAR-T2061-10mg10mg£225.00
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Quantity:
TAR-T2061-25mg25mg£349.00
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Quantity:
TAR-T2061-50mg50mg£544.00
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Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
APY0201 is a effective, highly specific, ATP-competitive PIKfyve inhibitor (IC50: 5.2 nM). It can interrupt the conversion of phosphatidylinositol 3-phosphate (PtdIns3P) to PtdIns(3, 5)P2.
CAS:
1232221-74-7
Formula:
C23H23N7O
Molecular Weight:
413.485
Pathway:
Immunology/Inflammation; PI3K/Akt/mTOR signaling
Purity:
0.9921
SMILES:
Cc1cccc(C=NNc2cc(N3CCOCC3)n3nc(cc3n2)-c2ccncc2)c1
Target:
PI3K; Interleukin

References

1. Hayakawa N, et al. Bioorg Med Chem. 2014 Jun 1;22(11):3021-9.