TargetMol

H4 Receptor antagonist 1

Product Code:
 
TAR-T5829
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T5829-1mg1mg£95.00
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TAR-T5829-2mg2mg£106.00
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TAR-T5829-5mg5mg£128.00
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TAR-T5829-1mL1 mL * 10 mM (in DMSO)£134.00
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TAR-T5829-10mg10mg£161.00
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TAR-T5829-25mg25mg£246.00
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TAR-T5829-50mg50mg£389.00
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TAR-T5829-100mg100mg£546.00
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Further Information

Bioactivity:
H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.
CAS:
848217-00-5
Formula:
C16H17ClN4O
Molecular Weight:
316.79
Pathway:
GPCR/G Protein; Neuroscience; Immunology/Inflammation
Purity:
0.98
SMILES:
CN1CCN(CC1)c1nc(C)nc2c3cc(Cl)ccc3oc12
Target:
Histamine Receptor

References

Cramp S , Dyke H J , Higgs C , et al. Identification and hit-to-lead exploration of a novel series of histamine H4 receptor inverse agonists[J]. Bioorganic & Medicinal Chemistry Letters, 2010, 20(8):2516-2519.