TargetMol

Selective PI3Kδ Inhibitor 1

Product Code:
 
TAR-T5831
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T5831-1mg1mg£158.00
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TAR-T5831-2mg2mg£201.00
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TAR-T5831-5mg5mg£328.00
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TAR-T5831-10mg10mg£458.00
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TAR-T5831-25mg25mg£704.00
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TAR-T5831-50mg50mg£938.00
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TAR-T5831-100mg100mg£1,259.00
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This product comes from: United States.
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Further Information

Bioactivity:
Selective PI3Kδ Inhibitor 1 is a PI3Kδ Inhibitor( IC50 = 0.9 nM).
CAS:
2088525-31-7
Formula:
C23H20FN7O
Molecular Weight:
429.459
Pathway:
PI3K/Akt/mTOR signaling
Purity:
0.98
SMILES:
Cn1nc(nc1C1(CC1)c1ccccc1)-c1cnc(N)c(n1)-c1ccc(C(N)=O)c(F)c1
Target:
PI3K

References

Terstiege I , Perry M , Petersen J , et al. Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K? inhibitors[J]. Bioorganic & medicinal chemistry letters, 2016, 27(3).