TargetMol

PROTAC ERR α ligand 2

Product Code:
 
TAR-T5835
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T5835-1mg1mg£119.00
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TAR-T5835-2mg2mg£141.00
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TAR-T5835-5mg5mg£189.00
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TAR-T5835-1mL1 mL * 10 mM (in DMSO)£201.00
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TAR-T5835-10mg10mg£229.00
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TAR-T5835-25mg25mg£389.00
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TAR-T5835-50mg50mg£550.00
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TAR-T5835-100mg100mg£755.00
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Further Information

Bioactivity:
PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist( IC50 : 5.67 nM)
CAS:
2306388-57-6
Formula:
C20H13F6NO4
Molecular Weight:
445.317
Pathway:
Endocrinology/Hormones
Purity:
0.98
SMILES:
COc1cc(C=C(/C#N)C(O)=O)ccc1OCc1ccc(cc1C(F)(F)F)C(F)(F)F
Target:
Estrogen Receptor/ERR; Estrogen/progestogen Receptor

References

Peng L , Zhang Z , Lei C , et al. Identification of New Small-Molecule Inducers of Estrogen-Related Receptor alpha (ERRa) Degradation[J]. ACS Medicinal Chemistry Letters, 2019, 10(5).