TargetMol

BMS-911543

Product Code:
 
TAR-T6790
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T6790-1mg1mg£111.00
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TAR-T6790-2mg2mg£128.00
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TAR-T6790-1mL1 mL * 10 mM (in DMSO)£161.00
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TAR-T6790-5mg5mg£164.00
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TAR-T6790-10mg10mg£225.00
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TAR-T6790-25mg25mg£389.00
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TAR-T6790-50mg50mg£547.00
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Further Information

Bioactivity:
BMS-911543 is a potent and selective inhibitor of JAK2 with IC50 of 1.1 nM, ~350-, 75- and 65-fold selective to JAK1, JAK3 and TYK2, respectively. Phase 1/2.
CAS:
1271022-90-2
Formula:
C23H28N8O
Molecular Weight:
432.532
Pathway:
Angiogenesis; Stem Cells; Tyrosine Kinase/Adaptors; Chromatin/Epigenetic; JAK/STAT signaling
Purity:
0.9998
SMILES:
CCn1c(cc2c1nc(Nc1cc(C)n(C)n1)c1ncn(C)c21)C(=O)N(C1CC1)C1CC1
Target:
Tyrosine Kinases; Histone Methyltransferase; JAK

References

Wan H, et al. ACS Med Chem Lett. 2015, 6(8):850-5.