TargetMol

ORY1001

Product Code:
 
TAR-T6922
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T6922-1mg1mg£114.00
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TAR-T6922-2mg2mg£132.00
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TAR-T6922-1mL1 mL * 10 mM (in DMSO)£180.00
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TAR-T6922-5mg5mg£180.00
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TAR-T6922-10mg10mg£268.00
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TAR-T6922-25mg25mg£452.00
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TAR-T6922-50mg50mg£629.00
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TAR-T6922-100mg100mg£864.00
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Quantity:
TAR-T6922-500mg500mg£1,661.00
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This product comes from: United States.
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Further Information

Bioactivity:
ORY-1001 (RG-6016) is an orally active and selective lysine-specific demethylase LSD1/KDM1A inhibitor, with high selectivity against related FAD dependent aminoxidases with IC50 of <20 nM.
CAS:
1431326-61-2
Formula:
C15H24Cl2N2
Molecular Weight:
303.27
Pathway:
Chromatin/Epigenetic
Purity:
0.9996
SMILES:
Cl.Cl.NC1CCC(CC1)N[C@@H]1C[C@H]1c1ccccc1
Target:
Histone Demethylase

References

Barbagallo C, Caltabiano R, Broggi G, et al. LncRNA LINC00518 Acts as an Oncogene in Uveal Melanoma by Regulating an RNA-Based Network. Cancers. 2020, 12(12): 3867 Barbagallo C, Caltabiano R, Broggi G, et al. LncRNA LINC00518 Acts as an Oncogene in Uveal Melanoma by Regulating an RNA-Based Network[J]. Cancers. 2020, 12(12): 3867 Maes T, et al. J Clin Oncol. 2013, 31, suppl; abstr. e13543. Lv S, Zhao X, Zhang E, et al. Lysine demethylase KDM1A promotes cell growth via FKBP8-BCL2 axis in hepatocellular carcinoma. Journal of Biological Chemistry. 2022: 102374.