TargetMol

Gabazine

Product Code:
 
TAR-T7622
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T7622-5mg5mg£108.00
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TAR-T7622-1mL1 mL * 10 mM (in DMSO)£112.00
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TAR-T7622-10mg10mg£128.00
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TAR-T7622-25mg25mg£185.00
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TAR-T7622-50mg50mg£289.00
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TAR-T7622-100mg100mg£462.00
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Quantity:
TAR-T7622-200mg200mg£600.00
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This product comes from: United States.
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Further Information

Bioactivity:
Gabazine is an antagonist of GABAA receptors (Ki : 74-150 nM)
CAS:
104104-50-9
Formula:
C15H18BrN3O3
Molecular Weight:
368.231
Pathway:
Neuroscience; Membrane transporter/Ion channel
Purity:
0.982
SMILES:
Br.COc1ccc(cc1)-c1ccc(=N)n(CCCC(O)=O)n1
Target:
GABA Receptor

References

Ueno S , Bracamontes J , Zorumski C , et al. Bicuculline and Gabazine Are Allosteric Inhibitors of Channel Opening of the GABA A Receptor[J]. The Journal of Neuroscience, 1997, 17(2):625-634. Chesnoy-Marchais, D. Persistent GABAA/C responses to gabazine, taurine and beta-alanine in rat hypoglossal motoneurons[J]. Neuroscience, 2016:S030645221630207X. Mendu S K , Amol B , Zhe J , et al. Different Subtypes of GABA-A Receptors Are Expressed in Human, Mouse and Rat T Lymphocytes[J]. PLoS ONE, 2012, 7(8):e42959-.