TargetMol

M4 mAChR agonist-1?

Product Code:
 
TAR-T9889
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
 

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CodeSizePrice
TAR-T9889-2mg2mg£102.00
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Quantity:
TAR-T9889-1mL1 mL * 10 mM (in DMSO)£122.00
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TAR-T9889-5mg5mg£122.00
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TAR-T9889-10mg10mg£148.00
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TAR-T9889-25mg25mg£213.00
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TAR-T9889-50mg50mg£303.00
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Quantity:
TAR-T9889-100mg100mg£414.00
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Quantity:
TAR-T9889-500mg500mg£849.00
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Further Information

Bioactivity:
M4 mAChR agonist-1 is an effective agonist of M4 mAChR (EC50 >10 μM).
CAS:
785705-53-5
Formula:
C14H18N4OS
Molecular Weight:
290.389
Pathway:
Neuroscience
Purity:
0.9825
SMILES:
CC1=C(C)C2=C(N=CN=C2S1)N1CCC(CC1)C(N)=O
Target:
AChR

References

Wood MR, et al. Discovery and optimization of a novel series of highly CNS penetrant M4 PAMs based on a 5,6-dimethyl-4-(piperidin-1-yl)thieno[2,3-d]pyrimidine core. Bioorg Med Chem Lett. 2016;26(13):3029-3033.