TargetMol

Cinacalcet metabolite M4

Product Code:
 
TAR-T10814
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T10814-1mL1 mL * 10 mM (in DMSO)£108.00
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TAR-T10814-5mg5mg£111.00
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TAR-T10814-10mg10mg£125.00
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TAR-T10814-25mg25mg£148.00
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TAR-T10814-50mg50mg£182.00
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TAR-T10814-100mg100mg£214.00
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TAR-T10814-200mg200mg£276.00
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TAR-T10814-500mg500mg£379.00
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Further Information

Bioactivity:
Cinacalcet metabolite M4 is a metabolite of Cinacalcet. Cinacalcet is an allosteric agonist of Ca receptor.
CAS:
104774-87-0
Formula:
C10H12F3N
Molecular Weight:
203.208
Pathway:
Metabolism; Membrane transporter/Ion channel
Purity:
0.9528
SMILES:
NCCCc1cccc(c1)C(F)(F)F
Target:
Calcium Channel

References

1. Kumar GN, et al. Metabolism and disposition of calcimimetic agent cinacalcet HCl in humans and animalmodels. Drug Metab Dispos. 2004 Dec;32(12):1491-500. 2. Bushinsky DA, et al. Effect of cinacalcet on urine calcium excretion and supersaturation in genetic hypercalciuric stone-forming rats. Kidney Int. 2006 May;69(9):1586-92.