TargetMol

GABAB receptor antagonist 1

Product Code:
 
TAR-T11350
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11350-5mg5mg£850.00
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TAR-T11350-50mg50mg£1,661.00
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TAR-T11350-100mg100mg£2,079.00
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Further Information

Bioactivity:
(E)-GABAB receptor antagonist 1 decreases GABA-induced IP3 (inositol trisphosphate) production with IC50 of 37.9 μM.GABAB receptor antagonist 1 is a selective and negative allosteric modulator of GABAB (γ-Aminobutyric acid) receptors.
CAS:
797-17-1
Formula:
C18H24O4
Molecular Weight:
304.386
Pathway:
Membrane transporter/Ion channel; Neuroscience
Purity:
0.98
SMILES:
CC(C)(C)c1cc(C=CC(=O)C(O)=O)cc(c1O)C(C)(C)C
Target:
GABA Receptor

References

1. Chen LH, et al. Discovery of a Negative Allosteric Modulator of GABAB Receptors. ACS Med Chem Lett. 2014 May 27;5(7):742-7.