TargetMol

sPLA2-X Inhibitor 31

Product Code:
 
TAR-T12990
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12990-5mg5mg£850.00
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TAR-T12990-50mg50mg£1,661.00
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Quantity:
TAR-T12990-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
sPLA2-X Inhibitor 31 is a selective inhibitor of secreted phospholipase A2 type X (sPLA2-X) (IC50s of 26 nM, 310 nM, and 2230 nM for sPLA2-X, sPLA2-IIa, and sPLA2-V, respectively).
CAS:
2241025-50-1
Formula:
C19H15F3N2O4
Molecular Weight:
392.334
Purity:
0.98
SMILES:
NC(=O)c1cc2ccc(OC(F)(F)F)cc2n1-c1cccc(CCC(O)=O)c1

References

1. Knerr L, et al. Discovery of a Series of Indole-2 Carboxamides as Selective Secreted Phospholipase A2 Type X(sPLA2-X) Inhibitors. ACS Med Chem Lett. 2018 Jun 23;9(7):594-599.