TargetMol

SSTR5 antagonist 2

Product Code:
 
TAR-T13022
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T13022-5mg5mg£930.00
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Quantity:
TAR-T13022-50mg50mg£1,821.00
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Quantity:
TAR-T13022-100mg100mg£2,319.00
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This product comes from: United States.
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Further Information

Bioactivity:
SSTR5 antagonist 2 is a highly potent, oral active and selective antagonist of somatostatin (receptor) subtype 5 (SSTR5),with potential to treat type 2 diabetes mellitus (T2DM).
CAS:
1254730-81-8
Formula:
C32H35FN2O5
Molecular Weight:
546.639
Purity:
0.98
SMILES:
CCOc1cc(CN2CCC3(CN(C(=O)C3)c3ccc(cc3)C(O)=O)CC2)cc(OCC)c1-c1ccc(F)cc1

References

1. Liu W, et al. Discovery and Pharmacology of a Novel Somatostatin Subtype 5 (SSTR5) Antagonist: Synergy with DPP-4 Inhibition. ACS Med Chem Lett. 2018 Sep 12;9(11):1082-1087.