TargetMol

VU0134992 hydrochloride

Product Code:
 
TAR-T13316
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T13316-2mg2mg£98.00
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TAR-T13316-5mg5mg£115.00
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TAR-T13316-1mL1 mL * 10 mM (in DMSO)£119.00
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TAR-T13316-10mg10mg£149.00
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TAR-T13316-25mg25mg£217.00
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TAR-T13316-50mg50mg£321.00
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TAR-T13316-100mg100mg£497.00
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Further Information

Bioactivity:
VU0134992 hydrochloride is the first subtype-preferring, orally active and selective blocker of Kir4.1 potassium channel pore(IC50 : 0.97 μM).
CAS:
1052515-91-9
Formula:
C20H32BrClN2O2
Molecular Weight:
447.84
Pathway:
Membrane transporter/Ion channel
Purity:
1
SMILES:
Cl.CC(C)c1ccc(OCC(=O)NC2CC(C)(C)NC(C)(C)C2)c(Br)c1
Target:
Potassium Channel

References

1. Kharade SV, et al. Discovery, Characterization, and Effects on Renal Fluid and Electrolyte Excretion of the Kir4.1 Potassium Channel Pore Blocker, VU0134992. Mol Pharmacol. 2018 Aug;94(2):926-937.