TargetMol

GS-9901

Product Code:
 
TAR-T15420
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T15420-5mg5mg£850.00
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Quantity:
TAR-T15420-50mg50mg£1,661.00
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Quantity:
TAR-T15420-100mg100mg£2,079.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
GS-9901 is a highly selective and orally active inhibitor of PI3Kδ (IC50: 1 nM). It also has the potential to treat rheumatoid arthritis.
CAS:
1640247-87-5
Formula:
C22H17ClFN9O
Molecular Weight:
477.89
Pathway:
PI3K/Akt/mTOR signaling
Purity:
0.98
SMILES:
Nc1nc(N)c(C#N)c(N[C@H](C2CC2)c2nc3c(F)ccc(Cl)c3c(=O)n2-c2cccnc2)n1
Target:
PI3K

References

1. Patel L, et al. Discovery of Orally Efficacious Phosphoinositide 3-Kinase ? Inhibitors with Improved Metabolic Stability. J Med Chem. 2016 Oct 13;59(19):9228-9242.