TargetMol

CDK4-IN-1

Product Code:
 
TAR-T2082
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T2082-5mg5mg£850.00
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Further Information

Bioactivity:
CDK4 inhibitor is a novel and specific CDK4/Cyclin D1 inhibitor with an IC50 of 10 nM; 1500 and 500 fold than CDK1/Cyclin B (IC50>15 uM) and CDK2/Cyclin A (IC50=5.265 uM) respectively.
CAS:
1256963-02-6
Formula:
C22H29ClN8
Molecular Weight:
440.98
Pathway:
Cell Cycle/Checkpoint
Purity:
0.98
SMILES:
CC(C)c1[nH]nc(Cl)c1-c1ccnc(Nc2ccc(cn2)N2CCC(CC2)N(C)C)n1
Target:
CDK

References

1. Cho YS, et al. J Med Chem. 2010 Nov 25;53(22):7938-57.