TargetMol

CGP 64213

Product Code:
 
TAR-T26995
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T26995-5mg5mg£1,091.00
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TAR-T26995-50mg50mg£2,143.00
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Quantity:
TAR-T26995-100mg100mg£2,801.00
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  • Further Information
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Further Information

Bioactivity:
CGP 64213 is a GABAb receptor agonist.
CAS:
200402-50-2
Formula:
C26H36IN2O7P
Molecular Weight:
646.459
Purity:
0.98
SMILES:
C[C@@H](NC[C@H](O)CP(O)(=O)CCCCCNC(=O)CCc1ccc(O)c(I)c1)c1cccc(c1)C(O)=O

References

1. Duthey B, Caudron S, Perroy J, Bettler B, Fagni L, Pin JP, Pr?zeau L. A single subunit (GB2) is required for G-protein activation by the heterodimeric GABA(B) receptor. J Biol Chem. 2002 Feb 1;277(5):3236-41. PubMed PMID: 11711539; PubMed Central PMCID: PMC2566549. 2. Calon F, Lavertu N, Lemieux AM, Morissette M, Goulet M, Grondin R, Blanchet PJ, B?dard PJ, Di Paolo T. Effect of MPTP-induced denervation on basal ganglia GABA(B) receptors: correlation with dopamine concentrations and dopamine transporter. Synapse. 2001 Jun 1;40(3):225-34. PubMed PMID: 11304760. 3. Calon F, Morissette M, Goulet M, Grondin R, Blanchet PJ, B?dard PJ, Di Paolo T. 125I-CGP 64213 binding to GABA(B) receptors in the brain of monkeys: effect of MPTP and dopaminomimetic treatments. Exp Neurol. 2000 May;163(1):191-9. PubMed PMID: 10785458. 4. Froestl W, Bettler B, Bittiger H, Heid J, Kaupmann K, Mickel SJ, Strub D. Ligands for the isolation of GABA(B) receptors [corrected] . Neuropharmacology. 1999 Nov;38(11):1641-6. Review. Erratum in: Neuropharmacology 1999 Dec;38(12):1921. PubMed PMID: 10587079.