TargetMol

DU-125530

Product Code:
 
TAR-T27215
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T27215-5mg5mg£1,091.00
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Quantity:
TAR-T27215-50mg50mg£2,143.00
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Quantity:
TAR-T27215-100mg100mg£2,801.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
DU-125530 is a 5-HT1A receptor antagonist.
CAS:
161611-99-0
Formula:
C23H26ClN3O5S
Molecular Weight:
491.99
Purity:
0.98
SMILES:
Clc1cc2OCCOc2c(c1)N1CCN(CCCCN2C(=O)c3ccccc3S2(=O)=O)CC1

References

1. Scorza MC, Llad?-Pelfort L, Oller S, Cort?s R, Puigdemont D, Portella MJ, P?rez-Egea R, Alvarez E, Celada P, P?rez V, Artigas F. Preclinical and clinical characterization of the selective 5-HT(1A) receptor antagonist DU-125530 for antidepressant treatment. Br J Pharmacol. 2012 Nov;167(5):1021-34. doi: 10.1111/j.1476-5381.2011.01770.x. PubMed PMID: 22050051; PubMed Central PMCID: PMC3492984. 2. Mos J, Van Hest A, Van Drimmelen M, Herremans AH, Olivier B. The putative 5-HT1A receptor antagonist DU125530 blocks the discriminative stimulus of the 5-HT1A receptor agonist flesinoxan in pigeons. Eur J Pharmacol. 1997 May 1;325(2-3):145-53. PubMed PMID: 9163561.