TargetMol

TPC-144

Product Code:
 
TAR-T28999
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T28999-5mg5mg£1,010.00
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TAR-T28999-50mg50mg£1,982.00
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TAR-T28999-100mg100mg£2,560.00
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This product comes from: United States.
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Further Information

Bioactivity:
TPC-144 is a potent and selective LSD1 inhibitor with a reversible inhibition mechanism. TPC-144 has antitumor activity in several human AML and SCLC cell lines and xenograft models.
CAS:
2098621-17-9
Formula:
C31H31F2N3O2
Molecular Weight:
515.605
Purity:
0.98
SMILES:
CC(C)(O)Cc1ccc(c(F)c1)-c1ccc(cc1-c1ccc(C#N)c(F)c1)C(=O)N1[C@H]2CC[C@@H]1C[C@H](N)C2

References

1. TPC-144, a novel reversible LSD1 inhibitor, exhibited strong antitumor activity in preclinical models of AML and SCLC A. Kawagishi, et al. European Journal of Cancer, December 2016Volume 69, Supplement 1, Pages S86?S87. doi: http://dx.doi.org/10.1016/S0959-8049(16)32853-2