TargetMol

WRC-0571

Product Code:
 
TAR-T29162
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T29162-5mg5mg£850.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T29162-50mg50mg£1,661.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T29162-100mg100mg£2,079.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
WRC-0571 is a highly potent, selective antagonist of A1 adenosine receptors.
CAS:
501667-77-2
Formula:
C17H26N6O
Molecular Weight:
330.436
Purity:
0.98
SMILES:
CC(C)N(C)c1nc2c(NC3CC4CC3CC4O)ncnc2n1C

References

1. Clark AN, Youkey R, Liu X, Jia L, Blatt R, Day YJ, Sullivan GW, Linden J, Tucker AL. A1 adenosine receptor activation promotes angiogenesis and release of VEGF from monocytes. Circ Res. 2007 Nov 26;101(11):1130-8. Epub 2007 Sep 27. PubMed PMID: 17901362. 2. Shryock JC, Ozeck MJ, Belardinelli L. Inverse agonists and neutral antagonists of recombinant human A1 adenosine receptors stably expressed in Chinese hamster ovary cells. Mol Pharmacol. 1998 May;53(5):886-93. PubMed PMID: 9584215. 3. Jin X, Shepherd RK, Duling BR, Linden J. Inosine binds to A3 adenosine receptors and stimulates mast cell degranulation. J Clin Invest. 1997 Dec 1;100(11):2849-57. PubMed PMID: 9389751; PubMed Central PMCID: PMC508491. 4. Auchampach JA, Jin X, Wan TC, Caughey GH, Linden J. Canine mast cell adenosine receptors: cloning and expression of the A3 receptor and evidence that degranulation is mediated by the A2B receptor. Mol Pharmacol. 1997 Nov;52(5):846-60. PubMed PMID: 9351976.