TargetMol

CPFPX

Product Code:
 
TAR-T31086
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T31086-5mg5mg£850.00
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Further Information

Bioactivity:
CPFPX is a highly selective radioactive ligand for the A1 adenosine receptor (A1AR).
CAS:
227205-79-0
Formula:
C16H23FN4O2
Molecular Weight:
321.387
Purity:
0.98
SMILES:
CCCn1c(=O)n(CCC[18F])c2nc([nH]c2c1=O)C1CCCC1

References

1. Kroll T, Elmenhorst D, Weisshaupt A, Beer S, Bauer A. Reproducibility of non-invasive a1 adenosine receptor quantification in the rat brain using [(18)F]CPFPX and positron emission tomography. Mol Imaging Biol. 2014 Oct;16(5):699-709. doi: 10.1007/s11307-014-0729-0. PubMed PMID: 24595700. 2. Elmenhorst D, Kroll T, Wedekind F, Weisshaupt A, Beer S, Bauer A. In vivo kinetic and steady-state quantification of 18F-CPFPX binding to rat cerebral A1 adenosine receptors: validation by displacement and autoradiographic experiments. J Nucl Med. 2013 Aug;54(8):1411-9. doi: 10.2967/jnumed.112.115576. PubMed PMID: 23740103. 3. Elmenhorst D, Meyer PT, Matusch A, Winz OH, Bauer A. Caffeine occupancy of human cerebral A1 adenosine receptors: in vivo quantification with 18F-CPFPX and PET. J Nucl Med. 2012 Nov;53(11):1723-9. doi: 10.2967/jnumed.112.105114. PubMed PMID: 22966134.