TargetMol

Panomifene

Product Code:
 
TAR-T33876
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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TAR-T33876-5mg5mg£603.00
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TAR-T33876-50mg50mg£1,821.00
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TAR-T33876-100mg100mg£2,319.00
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Further Information

Bioactivity:
Panomiphene (Gyki-13504, EGIS-5650) is an anti-estrogen drug that is a tamoxifen (TMX) analogue.
CAS:
77599-17-8
Formula:
C25H24F3NO2
Molecular Weight:
427.467
Purity:
0.98
SMILES:
OCCNCCOc1ccc(cc1)C(=C(/c1ccccc1)C(F)(F)F)c1ccccc1

References

Erd?lyi-T?th V, Gyergyay F, Sz?mel I, Pap E, Kralov?nszky J, Bojti E, Cs?rgo M, Drabant S, Klebovich I. Pharmacokinetics of panomifene in healthy volunteers at phase I/a study. Anticancer Drugs. 1997 Jul;8(6):603-9. PubMed PMID: 9300575. Monostory K, Jemnitz K, Vereczkey L, Czira G. Species differences in metabolism of panomifene, an analogue of tamoxifen. Drug Metab Dispos. 1997 Dec;25(12):1370-8. PubMed PMID: 9394026. Liu X, Shimizu M, Hiyama T. A facile stereocontrolled approach to CF3-substituted triarylethenes: synthesis of panomifene. Angew Chem Int Ed Engl. 2004 Feb 6;43(7):879-82. PubMed PMID: 14767964. Konno T, Daitoh T, Noiri A, Chae J, Ishihara T, Yamanaka H. A highly regio- and stereoselective carbocupration of fluoroalkylated internal alkynes: a short total synthesis of the antiestrogenic drug panomifene. Org Lett. 2004 Mar 18;6(6):933-6. PubMed PMID: 15012068.