TargetMol

AM-0902

Product Code:
 
TAR-T7430
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T7430-1mg1mg£98.00
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TAR-T7430-5mg5mg£132.00
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TAR-T7430-1mL1 mL * 10 mM (in DMSO)£139.00
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TAR-T7430-10mg10mg£156.00
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TAR-T7430-25mg25mg£249.00
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TAR-T7430-50mg50mg£417.00
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Quantity:
TAR-T7430-100mg100mg£584.00
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This product comes from: United States.
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Further Information

Bioactivity:
AM-0902 is a potent and specific TRPA1 antagonist (IC50s: 71/131 nM for rTRPA1 and hTRPA1).
CAS:
1883711-97-4
Formula:
C17H15ClN6O2
Molecular Weight:
370.8
Pathway:
Membrane transporter/Ion channel
Purity:
1
SMILES:
Cn1cnc2ncn(Cc3nc(CCc4ccc(Cl)cc4)no3)c(=O)c12
Target:
TRP/TRPV Channel

References

Schenkel LB, et al. Optimization of a Novel Quinazolinone-Based Series of Transient Receptor Potential A1 (TRPA1)Antagonists Demonstrating Potent in Vivo Activity. J Med Chem. 2016 Mar 24;59(6):2794-809.