TargetMol

Thalidomide-O-amido-C3-NH2 TFA

Product Code:
 
TAR-T7760
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T7760-5mg5mg£108.00
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TAR-T7760-10mg10mg£135.00
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TAR-T7760-25mg25mg£188.00
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TAR-T7760-50mg50mg£269.00
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TAR-T7760-100mg100mg£366.00
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TAR-T7760-200mg200mg£507.00
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Quantity:
TAR-T7760-500mg500mg£764.00
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Further Information

Bioactivity:
Thalidomide-O-amido-C3-NH2 TFA is a synthesized E3 ligase ligand-linker conjugate. Thalidomide-O-amido-C3-NH2 TFA incorporates the Thalidomide based cereblon ligand and a linker used in PROTAC technology.
CAS:
2022182-58-5
Formula:
C20H21F3N4O8
Molecular Weight:
502.403
Pathway:
PROTAC
Purity:
0.9847
SMILES:
OC(=O)C(F)(F)F.NCCCNC(=O)COc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12
Target:
Ligand for E3 Ligase|E3 Ligase Ligand-Linker Conjugate

References

Lohbeck J, et al. Practical synthesis of a phthalimide-based Cereblon ligand to enable PROTAC development. Bioorg Med Chem Lett. 2016 Nov 1;26(21):5260-5262.