TargetMol

CRT0066101 dihydrochloride

Product Code:
 
TAR-TQ0104
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
❮❯

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CodeSizePrice
TAR-TQ0104-1mg1mg£95.00
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TAR-TQ0104-5mg5mg£128.00
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TAR-TQ0104-1mL1 mL * 10 mM (in DMSO)£134.00
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TAR-TQ0104-10mg10mg£168.00
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TAR-TQ0104-25mg25mg£269.00
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TAR-TQ0104-50mg50mg£386.00
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Further Information

Bioactivity:
CRT0066101 dihydrochloride is an effective and selective PKD inhibitor (IC50s: 1, 2.5 and 2 nM for PKD1, 2, and 3).
CAS:
1883545-60-5
Formula:
C18H24Cl2N6O
Molecular Weight:
411.33
Pathway:
Metabolism; Cell Cycle/Checkpoint
Purity:
0.9985
SMILES:
Cl.Cl.CC[C@@H](N)CNc1ccnc(n1)-c1cc(ccc1O)-c1cnn(C)c1
Target:
Serine/threonin kinase

References

Harikumar KB, et al. A novel small-molecule inhibitor of protein kinase D blocks pancreatic cancer growth in vitro and in vivo. Mol Cancer Ther. 2010 May;9(5):1136-46.