TargetMol

bio-THZ1

Product Code:
 
TAR-T10546
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T10546-10mg10mg£1,916.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T10546-25mg25mg£3,854.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
bio-THZ1 is a biotinylated version of THZ1. THZ1 is a selective and irreversibly covalent CDK7 inhibitor (IC50: 3.2 nM).
CAS:
1604811-14-4
Formula:
C52H65ClN12O8S
Molecular Weight:
1053.68
Pathway:
Cell Cycle/Checkpoint
Purity:
0.98
SMILES:
[H][C@]12CS[C@@H](CCCCC(=O)NCCOCCOCCOCCNC(=O)NCCCN(C)CC=CC(=O)Nc3ccc(cc3)C(=O)Nc3cccc(Nc4ncc(Cl)c(n4)-c4c[nH]c5ccccc45)c3)[C@@]1([H])NC(=O)N2
Target:
CDK

References

1. Kwiatkowski N, et al. Targeting transcription regulation in cancer with a covalent CDK7 inhibitor. Nature. 2014 Jul 31;511(7511):616-20.