TargetMol

BRCA1-IN-2

Product Code:
 
TAR-T10601
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T10601-5mg5mg£390.00
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Quantity:
TAR-T10601-50mg50mg£1,629.00
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Quantity:
TAR-T10601-100mg100mg£2,432.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
BRCA1-IN-2 is a cell-permeable protein-protein interaction (PPI) inhibitor for BRCA1 (IC50: 0.31 μM; Kd: 0.3 μM). It has antitumor activities via the disruption of BRCA1 (BRCT)2/protein interactions.
CAS:
1622262-55-8
Formula:
C26H33N4O7P
Molecular Weight:
544.545
Purity:
0.98
SMILES:
OP(O)(=O)OC[C@H](NC(=O)CCc1c[nH]c2ccccc12)C(=O)NCC(=O)NCCCCc1ccccc1

References

1. Na Z, et al. Protein-Protein Interaction Inhibitors of BRCA1 Discovered Using Small Molecule Microarrays. Methods Mol Biol. 2017;1518:139-156.