TargetMol

Dihydromunduletone

Product Code:
 
TAR-T11044
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
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TAR-T11044-5mg5mg£1,552.00
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Further Information

Bioactivity:
Dihydromunduletone (DHM) is a carotenoid derivative and selective strong adhesion G protein-coupled receptor (aGPCR) (GPR56 and GPR114/ADGRG5) antagonists, does not inhibit GPR110 or class A GPCR, IC 50 20.9μM.
CAS:
674786-20-0
Formula:
C25H28O6
Molecular Weight:
424.493
Pathway:
GPCR/G Protein; Endocrinology/Hormones
Purity:
0.98
SMILES:
COc1c(CC(=O)c2cc3CC(O)C(C)(C)Oc3cc2O)ccc2OC(C)(C)C=Cc12
Target:
GPR

References

1. Hannah M. Stoveken, et al. Dihydromunduletone Is a Small-Molecule Selective Adhesion G Protein?Coupled Receptor Antagonist. Mol Pharmacol. 2016 Sep; 90(3): 214?224.