TargetMol

Rivanicline hemioxalate

Product Code:
 
TAR-T12738
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12738-500mg500mg£1,495.00
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Further Information

Bioactivity:
Rivanicline hemioxalate is an agonist of neuronal nicotinic receptor, showing high selectivity for the α4β2 subtype (Ki=26 nM).
CAS:
T12738
Formula:
C11H15N2O2
Molecular Weight:
207.23
Purity:
0.98
SMILES:
CNCC/C=C/C1=CC=CN=C1.OC(C(O)=O)=O.[0.5]

References

1. Bencherif M, et al. RJR-2403: a nicotinic agonist with CNS selectivity I. In vitro characterization. J Pharmacol Exp Ther. 1996 Dec;279(3):1413-21. 2. Lippiello PM, et al. RJR-2403: a nicotinic agonist with CNS selectivity II. In vivo characterization. J Pharmacol Exp Ther. 1996 Dec;279(3):1422-9. 3. Damaj MI, et al. Antinociceptive and pharmacological effects of metanicotine, a selective nicotinic agonist. J Pharmacol Exp Ther. 1999 Oct;291(1):390-8.