TargetMol

Tertiapin LQ

Product Code:
 
TAR-TP2113
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
 

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CodeSizePrice
TAR-TP2113-10mg10mg£475.00
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Further Information

Bioactivity:
Blocker of Kir1.1 channels; displays >250-fold selectivity for Kir1.1 (Kd values are 1.1, 274 and 361 nM for Kir1.1, Kir3.1/3.2 and Kir3.1/3.4 respectively). Derivative of tertiapin-Q.
CAS:
TP2113
Formula:
C106H179N33O24S4
Molecular Weight:
2428.03
Purity:
0.98
SMILES:
0

References

Ramu et al (2008) Engineered specific and high-affinity inhibitor for a subtype of inward-rectifier K+ channels. Proc.Natl.Acad.Sci.USA 105 10774 PMID: