TargetMol

RI-STAD 2

Product Code:
 
TAR-TP2129
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
 

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CodeSizePrice
TAR-TP2129-10mg10mg£1,466.00
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Further Information

Bioactivity:
AKAP disruptor. Selectively binds PKA-RI with high affinity (KD values are 6.2 and 12.1 nM for the RIα and β subunits, respectively) and blocks its interaction with AKAP. Inhibits type I PKA-mediated phosphorylation in live cells. Cell permeable.
CAS:
TP2129
Formula:
C109H181N25O35
Molecular Weight:
2401.75
Purity:
0.98
SMILES:
0

References

Wang et al (2015) PKA-type I selective constrained peptide disruptors of AKAP complexes. ACS Chem.Biol. 10 1502 PMID: