TargetMol

(R)-PS210

Product Code:
 
TAR-T12639
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
❮❯

No additional charges, what you see is what you pay! *

CodeSizePrice
TAR-T12639-50mg50mg£870.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T12639-100mg100mg£1,364.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
Prices exclude any Taxes / VAT
How to order with us   Contact us
Stay in control of your spending. These prices have no additional charges, not even shipping!
* Rare exceptions are clearly labelled (only 0.14% of items!).
Multibuy discounts available! Contact us to find what you can save.
This product comes from: United States.
Typical lead time: 10-14 working days.
Contact us for more accurate information.
  • Further Information
  • Documents
  • References
  • Show All

Further Information

Bioactivity:
(R)-PS210, the R enantiomer of PS210 is a substrate-selective allosteric PDK1 activator with an (AC50 of 1.8 μM).
CAS:
1410101-89-1
Formula:
C19H15F3O5
Molecular Weight:
380.319
Purity:
0.98
SMILES:
OC(=O)C([C@@H](CC(=O)c1ccc(cc1)C(F)(F)F)c1ccccc1)C(O)=O

References

1. Wilhelm A, et al. 2-(3-Oxo-1,3-diphenylpropyl)malonic?acids?as?potent?allosteric?ligands?of the?PIF?pocket?of?phosphoinositide-dependent?kinase-1:?development?and?prodrug?concept.J Med Chem.?2012 Nov 26;55(22):9817-30.